Small molecule FGF receptor inhibitors block FGFR-dependent urothelial carcinoma growth in vitro and in vivo
Publication date
2011Keyword
Animals;Apoptosis; Drug effects;
Benzimidazoles; Therapeutic use;
Blotting; Western;
Carcinoma; Transitional cell; Metabolism; Pathology; Prevention & control;
Cell cycle;
Cell proliferation;
Cells; Cultured;
Humans;
Immunoenzyme techniques;
Male;
Mice;
Inbred BALB C;
Mutation; Genetics;
Phosphorylation;
Protein-Tyrosine Kinases; Antagonists & inhibitors;
Pyrimidines; Therapeutic use;
Pyrroles;
Quinolones;
Receptor; Fibroblast growth factor; Type 1/antagonists & inhibitors; Metabolism;
Receptor, Fibroblast growth factor, Type 3/antagonists & inhibitors; Metabolism;
Urinary Bladder Neoplasms; Prevention & control;
Urothelium;
Xenograft model antitumor assays;
REF 2014